A blog founded by Teddy Zartler and run by Dan Erlanson for Fragment-based Drug Discovery devotees to discuss non-confidential issues regarding fragments.

Joined February 2019
Strategies for covalency: @VividionRx recognize covalent potential on inflammasome target NLRP3, scan proteome to find cryptic site, assess promiscuity, improve selectivity, and present a chemical probe in @BrJPharmacol practicalfragments.blogspot.…
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